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Article Abstract
Herein, we present an efficient and feasible strategy for direct C-H fluorination and heteroarylation of oxindoles on the C-3 position having a C(sp)-H bond with quinoxalin-2(1)-ones based on a radical coupling reaction Selectfluor, a bifunctional reagent, as both the oxidant and fluorine source. This methodology provides a potential protocol to obtain 3-heteroaryl 3-fluorooxindoles in medium to excellent yields.
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