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Article Abstract
It is universally acknowledged that ligands can improve the reaction activity to simplify the reaction operating conditions and enrich the applicability of the reaction. Therefore, we developed -octylglycine ligand-accelerated Pd-catalyzed -arylation of benzoic acids under mild conditions with just 6 h; moreover, this -octylglycine ligand was successfully implemented to carboxyl-directed Pd-catalyzed β-C(sp)-H arylation and arylation of phenylacetic acids under mild conditions.
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