Article Synopsis

  • New variants of SARS-CoV-2 are prolonging the COVID-19 pandemic, prompting research into potent inhibitors.
  • A unique homotrimeric miniprotein inhibitor called TRI2-2 was developed to effectively neutralize multiple variants, outperforming existing monoclonal antibodies.
  • TRI2-2 showed protective effects against SARS-CoV-2 in mice and may offer a therapeutic strategy that resists viral mutations and reduces autoimmune risks compared to other options.

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Article Abstract

New variants of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) continue to arise and prolong the coronavirus disease 2019 (COVID-19) pandemic. Here, we used a cell-free expression workflow to rapidly screen and optimize constructs containing multiple computationally designed miniprotein inhibitors of SARS-CoV-2. We found the broadest efficacy was achieved with a homotrimeric version of the 75-residue angiotensin-converting enzyme 2 (ACE2) mimic AHB2 (TRI2-2) designed to geometrically match the trimeric spike architecture. Consistent with the design model, in the cryo-electron microscopy structure TRI2-2 forms a tripod at the apex of the spike protein that engaged all three receptor binding domains simultaneously. TRI2-2 neutralized Omicron (B.1.1.529), Delta (B.1.617.2), and all other variants tested with greater potency than the monoclonal antibodies used clinically for the treatment of COVID-19. TRI2-2 also conferred prophylactic and therapeutic protection against SARS-CoV-2 challenge when administered intranasally in mice. Designed miniprotein receptor mimics geometrically arrayed to match pathogen receptor binding sites could be a widely applicable antiviral therapeutic strategy with advantages over antibodies in greater resistance to viral escape and antigenic drift, and advantages over native receptor traps in lower chances of autoimmune responses.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC9258422PMC
http://dx.doi.org/10.1126/scitranslmed.abn1252DOI Listing

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