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Article Abstract

Dirhodium(II) complex-catalyzed [3 + 2] reactions between -arylaminocyclopropanes and alkyne derivatives are described. The cycloaddition products proved to be versatile synthetic intermediates. -Cyclic β-amino acids and derivatives thereof can be conveniently synthesized using this cycloaddition protocol.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6404392PMC
http://dx.doi.org/10.3762/bjoc.15.48DOI Listing

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