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Article Abstract
We describe the impact of proline modifications, in our tetracyclic-indole based series of nonstructural protein 5A (NS5A) inhibitors, to their replicon profiles. This work identified NS5A inhibitors with an improved and flattened resistance profiles.
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| http://dx.doi.org/10.1016/j.bmcl.2016.08.097 | DOI Listing |
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